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TAK-779

Glpbio
Catalog No:GC37724-10mM (in 1mL DMSO) CAS No.:229005-80-5 MDLNo: Brand:Glpbio purity: 特性: Purpose:TAK-779 是一種有效的,選擇性的,非肽類 CCR5 和 CXCR3 拮抗劑,對 CCR5 的 Ki 值為 1.1 nM,同時可以有效地,選擇性地抑制 R5 HIV-1,在 MAGI-CCR5 細胞中,EC50 和 EC90 值分別為 1.2 nM 和 5.7 nM。DMSO: ≥ 25 mg/mL (47.07 mM); H2O: 16.66 mg/mL (31.37 mM and warming)
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